The structure of pure liquid water and solvent effects on the cis-trans isomerization of a model peptidic fragment, N-methylacetamide: ab initio and empirical model simulation studies



Dr. Yves MANTZ

Department of Chemistry and Applied Biosciences ETH Zurich CH-6900 Lugano, Switzerland


Lundi 22 mai 2006, 11 heures
Salle RAPHAEL 1 - site d'Ivry-sur-Seine

Liquid water's structure is important to understand and is currently a vigorous topic of debate in the literature. In this presentation, structural correlations in liquid water are systematically examined using increasingly realistic theoretical models, including empirical rigid, empirical polarizable, empirical flexible with classical and quantum nuclei, and ab initio (DFT-BLYP) with classical nuclei at 300 and 353 K and quantum nuclei at 300 K.
The results obtained from well-converged Car-Parrinello MD and MD simulations support a (traditional) tetrahedral model of liquid water and provide a useful benchmark for the study of solvated N-methylacetamide (NMA), a simple molecular model of the peptide linkage in proteins. Because of its small size, NMA is amenable to study by high resolution/accuracy experimental and theoretical techniques that are not easily applicable to large systems. Two distinctly different theoretical descriptions, an ab initio (DFT-BLYP) and an empirical (CHARMM22) model, of NMA in explicit water solvent are employed to characterize the solvent structure at equilibrium and changes in solvation structure accompanying the cis-trans isomerization of NMA. Additionally, the thermodynamic, structural, and electronic properties of NMA along a preselected isomerization pathway, i.e., the torsional twist angle about the peptidic C(O)-N bond, are probed by performing both umbrella-sampling CPMD and MD as well as static calculations. An electronic restructuring of the peptide bond is revealed using state-of-the-art analysis tools, namely ELF and Wannier functions, shedding further light on (changes in) the peptide partial-double bond in proteins.